HIF/HIF Prolyl-Hydroxylase Inhibitors

HIF-1α

HIF-1α

HIF-1α
HIF-1β

HIF-1α

HIF-1α, IC₅₀: .55 μM ([1])

HIF-1α, Kd: 14.5 μM
HIF-2α, Kd: 10.2 μM

HIF-1α, IC₅₀: 4.86 μM

HIF-1α, Kd: 65 μM
HIF-2α, Kd: 123 μM

HIF-1α